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3dmolformer: A dual-channel framework for structure-based drug discovery.arXiv preprint arXiv:2502.05107, 2025a

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cs.LG 1

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2026 1

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Fine-tuning Pocket-Aware Diffusion Models via Denoising Policy Optimization

cs.LG · 2026-05-17 · unverdicted · novelty 6.0

DEPPA reformulates the denoising process of pocket-aware diffusion models as a multi-step MDP and applies RL fine-tuning with a coarse scheduler to optimize ligands for binding affinity, drug-likeness, synthesizability and diversity on CrossDocked2020.

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  • Fine-tuning Pocket-Aware Diffusion Models via Denoising Policy Optimization cs.LG · 2026-05-17 · unverdicted · none · ref 7

    DEPPA reformulates the denoising process of pocket-aware diffusion models as a multi-step MDP and applies RL fine-tuning with a coarse scheduler to optimize ligands for binding affinity, drug-likeness, synthesizability and diversity on CrossDocked2020.