TACK dataset enables scaffold-based evaluation showing classical ML methods outperform a domain-specific GNN for PROTAC activity prediction, with potency far more predictable than maximum degradation.
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TACK: A statistical evaluation of degradation activity on a novel TArgeting Chimeras Knowledge dataset
TACK dataset enables scaffold-based evaluation showing classical ML methods outperform a domain-specific GNN for PROTAC activity prediction, with potency far more predictable than maximum degradation.